Cyclic Enamine synthesis

Inexpensive Multigram-Scale Synthesis of Cyclic Enamines and 3-*N* Spirocyclopropyl Systems

Cyclic enamines are important synthons for many synthetic and pharmacological targets. Here, we report an inexpensive, catalyst-free, multigram-scale synthesis for cyclic enamines with exocyclic double bonds and four- to seven-membered rings. This …

Lipidated Spirocyclopropyls

Synthesis of spirocyclic systems, cyclic enamines, and their conjugation to lipids